SCHEMBL8320472

SCHEMBL8320472

Cn1nc(C(=O)NC2CC3CC4CC(C2)N3C/C4=N\O)c2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.66
CYP3A4 P08684 1/20 0.66
TSHR P16473 1/20 0.66
MAPK1 P28482 1/20 0.66
HSD17B10 Q99714 1/20 0.66
HTR3A P46098 12/20 0.63
HTR3E A5X5Y0 1/20 0.63
SLC22A2 O15244 1/20 0.63
HTR3B O95264 1/20 0.63
CHRNB2 P17787 1/20 0.63
CHRNA3 P32297 1/20 0.63
CHRNA4 P43681 1/20 0.63
KCNH2 Q12809 1/20 0.63
HTR3D Q70Z44 1/20 0.63
HTR3C Q8WXA8 1/20 0.63
SLC47A1 Q96FL8 1/20 0.63
KDM4E B2RXH2 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8320476 1.00 ALDH1A1 (0.66) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8323114 1.00 ALDH1A1 (0.66) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8320481 1.00 ALDH1A1 (0.66) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8321339 0.87 ALDH1A1 (0.69) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8322383 0.87 ALDH1A1 (0.69) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8327265 0.87 ALDH1A1 (0.69) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL8318653 0.84 ALDH1A1 (0.66) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL9680622 0.80 ALDH1A1 (0.76) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL9680628 0.80 ALDH1A1 (0.76) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL9485783 0.80 ALDH1A1 (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0518767-A2 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS INC. (US) 1992-12-16 EP claimed
JP-5202044-A None JP disclosed
US-5955470-A Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS, INC. (US) 1999-09-21 US disclosed
JP-H05202044-A DERIVATIVE OF AMIDE ANALOG OF CERTAIN METHANO BRIDGED QUINOLIZINE MERRELL DOW PHARMACEUT INC 1993-08-10 JP disclosed
EP-0517984-A1 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL DOW PHARMACEUTICALS INC. (US) 1992-12-16 EP disclosed
EP-0518767-A2 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS INC. (US) 1992-12-16 EP disclosed