SCHEMBL9680628

SCHEMBL9680628

Cn1nc(C(=O)NC2CC3C[C@H]4CCN3[C@@H](C2)C4)c2ccccc21

nearest known ligand 0.76

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.76
CYP3A4 P08684 1/20 0.76
TSHR P16473 1/20 0.76
MAPK1 P28482 1/20 0.76
HSD17B10 Q99714 1/20 0.76
HTR3A P46098 11/20 0.72
HTR3E A5X5Y0 1/20 0.72
SLC22A2 O15244 1/20 0.72
HTR3B O95264 1/20 0.72
CHRNB2 P17787 1/20 0.72
CHRNA3 P32297 1/20 0.72
CHRNA4 P43681 1/20 0.72
KCNH2 Q12809 1/20 0.72
HTR3D Q70Z44 1/20 0.72
HTR3C Q8WXA8 1/20 0.72
SLC47A1 Q96FL8 1/20 0.72
KDM4E B2RXH2 1/20 0.67
HTR4 Q13639 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9680622 1.00 ALDH1A1 (0.76) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL9485783 0.86 ALDH1A1 (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL30596797 0.86 ALDH1A1 (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL445223 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL34178 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL13660190 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL4109977 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL4890 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL16642163 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL13287290 0.84 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0517984-A1 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL DOW PHARMACEUTICALS INC. (US) 1992-12-16 EP disclosed
EP-0518767-A2 Derivatives of amide analogs of certain methano bridged quinolizines MERRELL PHARMACEUTICALS INC. (US) 1992-12-16 EP disclosed