SCHEMBL8320601

SCHEMBL8320601

O=C(I)C1CCCN(C(=O)Nc2ccc(Cl)cc2)C1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.58
MAPT P10636 2/20 0.58
RAB9A P51151 2/20 0.58
LMNA P02545 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
NPC1 O15118 1/20 0.58
NFKB1 P19838 1/20 0.58
NFKB2 Q00653 1/20 0.58
RELA Q04206 1/20 0.58
POLB P06746 1/20 0.58
ALDH1A1 P00352 1/20 0.55
ALOX5 P09917 1/20 0.53
RHOA P61586 4/20 0.51
HPGD P15428 2/20 0.51
HTT P42858 1/20 0.51
RHOC P08134 1/20 0.51
CCR2 P41597 1/20 0.50
KCNH2 Q12809 1/20 0.50
CYP3A4 P08684 1/20 0.50
MEN1 O00255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL77309 0.88 MAPT (0.63) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL13234925 0.80 RAB9A (0.70) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL10596224 0.78 MAPT (0.69) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL13691562 0.78 MAPT (0.88) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL4198615 0.77 NPC1 (0.59) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL7298745 0.75 HPGD (0.69) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL27979652 0.75 CA12 (0.71) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL14414045 0.74 CCR2 (0.59) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL1574534 0.74 TP53 (0.57) TP53MAPTRAB9ALMNASMN1; SMN2
SCHEMBL1575212 0.74 TP53 (0.57) TP53MAPTRAB9ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087646-A2 PYRROLIDINO-1,2-DICARBOXY-1-(PHENYLAMIDE)-2-(4-(3-OXO-MORPHOLINO-4-YL)-PHENYLAMIDE) DERIVATIVES AND RELATED COMPOUNDS FOR USE AS INHIBITORS OF COAGULATION FACTOR XA IN THE TREATMENT OF THROMBO-EMBOLIC DISEASES MERCK PATENT GMBH (DE) 2004-10-14 WO disclosed