SCHEMBL8320939

SCHEMBL8320939

Cc1nnc2n1-c1ncccc1C(c1ccc(Cl)cc1)=NN2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.43
AKT1 P31749 1/20 0.38
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 1/20 0.34
GABRA1 P14867 1/20 0.34
HPGD P15428 1/20 0.34
CNR1 P21554 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
OPRK1 P41145 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
BRD2 P25440 1/20 0.34
BRD3 Q15059 1/20 0.34
POLB P06746 2/20 0.33
MAPT P10636 1/20 0.33
AVPR1A P37288 1/20 0.32
CCKBR P32239 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318668 0.81 BRD4 (0.59) BRD4LMNAGABRA1HPGDCNR1
SCHEMBL9886480 0.75 BRD4 (0.41) BRD4AKT1NPC1RAB9AKMT2A
SCHEMBL8317643 0.75 BRD4 (0.43) BRD4KMT2ALMNAGABRA1HPGD
SCHEMBL21847194 0.75 BRD4 (0.39) BRD4LMNAGABRA1HPGDCNR1
SCHEMBL17479961 0.74 BRD4 (0.42) BRD4AKT1NPC1RAB9AKMT2A
SCHEMBL8316669 0.72 OPRK1 (0.61) BRD4LMNAGABRA1HPGDCNR1
Bromide SCHEMBL8319843 0.71 OPRK1 (0.60) BRD4LMNAGABRA1HPGDCNR1
SCHEMBL8319224 0.71 BRD4 (0.46) BRD4AKT1BRD2BRD3
SCHEMBL8317008 0.70 OPRK1 (0.48) BRD4OPRK1BRD2BRD3
SCHEMBL8323556 0.70 BRD4 (0.54) BRD4LMNAGABRA1HPGDCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934940-A1 CYTOKINE PRODUCTION INHIBITORS, TRIAZEPINE COMPOUNDS, AND INTERMEDIATES THEREOF Japan Tobacco Inc. (JP) 1999-08-11 EP disclosed