SCHEMBL8322831

SCHEMBL8322831

NC12C=CC=CC1CN(c1cc3c(cc1F)c(=O)c(OC(=O)O)cn3[C@@H]1C[C@@H]1F)C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 4/20 0.35
LMNA P02545 3/20 0.35
HPGD P15428 3/20 0.35
HSD17B10 Q99714 3/20 0.35
CYP1A2 P05177 1/20 0.35
TOP2A P11388 1/20 0.35
CYP2C9 P11712 1/20 0.35
TOP2B Q02880 1/20 0.35
MAPT P10636 1/20 0.34
TOP1 P11387 1/20 0.32
PIK3CG P48736 7/20 0.31
CYP3A4 P08684 1/20 0.31
PIK3CD O00329 5/20 0.31
PIK3R1 P27986 5/20 0.31
PIK3CA P42336 5/20 0.31
DRD3 P35462 1/20 0.30
PRKD3 O94806 1/20 0.30
PIM1 P11309 1/20 0.30
GSK3A P49840 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323758 0.90 KDM4E (0.45) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8925001 0.88 ALDH1A1 (0.45) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8925004 0.88 ALDH1A1 (0.45) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8925008 0.86 KDM4E (0.36) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8323426 0.85 CYP3A4 (0.34) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL8323544 0.85 KDM4E (0.47) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8321532 0.85 ALDH1A1 (0.34) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8321538 0.84 EPHA2 (0.39) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8320645 0.83 ALDH1A1 (0.41) ALDH1A1CYP2C9CYP3A4
SCHEMBL8318803 0.83 ALDH1A1 (0.41) ALDH1A1CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705828-B1 Quinolone- and naphthyridone carboxylic acid derivatives as antibacterial agents BAYER AG (DE) 1999-12-01 EP disclosed
EP-0705828-A1 Quinolone- and naphthyridone carboxylic acid derivatives as antibacterial agents BAYER AG (DE) 1996-04-10 EP disclosed