SCHEMBL8322835

SCHEMBL8322835

O=C(O)c1cnc(CCc2ccccc2OCc2ccccc2)[nH]c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 4/20 0.52
KDM4A O75164 4/20 0.52
KDM4D Q6B0I6 4/20 0.52
HIF1AN Q9NWT6 4/20 0.52
KDM5B Q9UGL1 4/20 0.52
KDM2A Q9Y2K7 4/20 0.52
KDM3B Q7LBC6 3/20 0.52
HTR1A P08908 2/20 0.51
DRD2 P14416 2/20 0.51
PTGER1 P34995 1/20 0.49
PTGER4 P35408 1/20 0.49
PTGER3 P43115 1/20 0.49
PTGER2 P43116 1/20 0.49
ABCB1 P08183 2/20 0.48
DAO P14920 1/20 0.48
BRS3 P32247 3/20 0.47
PDE9A O76083 1/20 0.46
PDE1A P54750 1/20 0.46
PDE1B Q01064 1/20 0.46
PDE1C Q14123 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8320061 0.87 ALDH1A1 (0.53) HTR1ADRD2ABCB1DAOPDE9A
SCHEMBL8327202 0.82 ALDH1A1 (0.55) HTR1ADRD2PTGER1
SCHEMBL8326795 0.81 HTR1A (0.54) KDM6BKDM4AKDM4DHIF1ANKDM5B
SCHEMBL8327188 0.81 HTR1A (0.47) HTR1ADRD2ABCB1DAOPDE9A
SCHEMBL8321604 0.75 HTR1A (0.49) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8677419 0.74 HTR1A (0.54) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8674773 0.74 HTR1A (0.60) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8320867 0.74 ABCB1 (0.52) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8675205 0.73 PTGER1 (0.71) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8675521 0.73 PTGER1 (0.67) HTR1ADRD2PTGER1PTGER4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed