SCHEMBL8323407

SCHEMBL8323407

CSc1c(C#N)/c(=N/C(=O)Nc2ccccc2)n(C)c(=S)n1-c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
GRIA2 P42262 2/20 0.38
GRIA4 P48058 2/20 0.38
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
KDM4E B2RXH2 6/20 0.35
HPGD P15428 3/20 0.35
GAA P10253 3/20 0.35
TOP2A P11388 2/20 0.35
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
USP2 O75604 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323410 1.00 ALDH1A1 (0.39) ALDH1A1TSHRHSD17B10TAS1R3TAS1R1
SCHEMBL8327882 0.89 GRIA2 (0.43) ALDH1A1TSHRHSD17B10TAS1R3TAS1R1
SCHEMBL8328635 0.87 GRIA4 (0.38) ALDH1A1TSHRHSD17B10GRIA2GRIA4
SCHEMBL8328629 0.87 GRIA4 (0.38) ALDH1A1TSHRHSD17B10GRIA2GRIA4
SCHEMBL8328148 0.86 GRIA4 (0.41) ALDH1A1TSHRHSD17B10GRIA2GRIA4
SCHEMBL8328146 0.86 GRIA4 (0.41) ALDH1A1TSHRHSD17B10GRIA2GRIA4
SCHEMBL8327668 0.84 GRIA2 (0.41) ALDH1A1TSHRHSD17B10TAS1R3TAS1R1
SCHEMBL8327673 0.84 GRIA2 (0.41) ALDH1A1TSHRHSD17B10TAS1R3TAS1R1
SCHEMBL8328436 0.84 ALDH1A1 (0.38) ALDH1A1TSHRHSD17B10TAS1R3TAS1R1
SCHEMBL8328438 0.84 ALDH1A1 (0.38) ALDH1A1TSHRHSD17B10TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed