SCHEMBL8323696

SCHEMBL8323696

C[S+]([O-])c1ccc(-c2cnn(-c3ccc(F)c(F)c3)c(=O)c2OCCC(C)(C)O)cc1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.32
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8289110 0.88 MCHR1 (0.42) MCHR1
SCHEMBL14516861 0.87 MCHR1 (0.42) MCHR1PTGS2FFAR4
SCHEMBL221377 0.87 PTGS2 (0.43) PTGS1PTGS2
SCHEMBL29366997 0.87 PTGS2 (0.43) PTGS1PTGS2
SCHEMBL4197238 0.86 PTGS2 (0.41) PTGS1PTGS2
SCHEMBL4185476 0.86 PTGS2 (0.34) MCHR1PTGS2
SCHEMBL19953615 0.85 PTGS2 (0.36) PTGS1PTGS2
SCHEMBL17364528 0.85 NPBWR1 (0.34) MCHR1FFAR4
SCHEMBL2606110 0.83 NPBWR1 (0.33) MCHR1
SCHEMBL12052331 0.83 MCHR1 (0.33) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004060366-A1 A METHOD FOR THE TREATMENT, PREVENTION, OR INHIBITION OF A CNS DISORDER AND/OR PAIN AND INFLAMMATION USING A COMBINATION OF DULOXETINE, VENLAFAXINE OR ATOMOXETINE AND A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR AND COMPOSITIONS THEREOF PHARMACIA CORPORATION (US) 2004-07-22 WO disclosed