SCHEMBL8324262

SCHEMBL8324262

N#Cc1ccc(N(Cc2cc(F)c(F)cc2F)c2cncnc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.40
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
CYP3A4 P08684 1/20 0.38
GRM5 P41594 2/20 0.36
VNN1 O95497 1/20 0.35
STS P08842 3/20 0.35
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326800 0.87 CYP19A1 (0.44) CYP19A1NOS3NOS1NOS2GRM5
SCHEMBL8325621 0.86 CYP19A1 (0.44) CYP19A1NOS3NOS1NOS2CYP3A4
SCHEMBL8327043 0.86 CYP19A1 (0.45) CYP19A1CYP3A4VNN1STS
SCHEMBL27282324 0.84 EGLN2 (0.38) CYP19A1NOS3NOS1NOS2CYP3A4
SCHEMBL8327987 0.80 CYP19A1 (0.42) CYP19A1VNN1STS
SCHEMBL6063814 0.80 CYP19A1 (0.38) CYP19A1GRM5VNN1
SCHEMBL8328066 0.79 CYP19A1 (0.44) CYP19A1STS
SCHEMBL30262487 0.79 CYP19A1 (0.37) CYP19A1NOS3NOS1NOS2CYP3A4
SCHEMBL28922397 0.79 CYP19A1 (0.46) CYP19A1STS
SCHEMBL8323103 0.78 ESR1 (0.49) CYP19A1VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed