SCHEMBL28922397

SCHEMBL28922397

N#Cc1ccc(N(Cc2ccc(C#N)c(F)c2)c2cncnc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.46
KDM1A O60341 1/20 0.45
CYP11B1 P15538 4/20 0.41
CYP11B2 P19099 4/20 0.41
STS P08842 2/20 0.40
TRPV4 Q9HBA0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327043 0.90 CYP19A1 (0.45) CYP19A1KDM1ASTS
SCHEMBL8329384 0.87 CYP19A1 (0.43) CYP19A1CYP11B1CYP11B2STS
SCHEMBL8327987 0.84 CYP19A1 (0.42) CYP19A1CYP11B1CYP11B2STS
SCHEMBL8328066 0.84 CYP19A1 (0.44) CYP19A1CYP11B1CYP11B2STS
SCHEMBL8323103 0.83 ESR1 (0.49) CYP19A1KDM1ACYP11B1CYP11B2
SCHEMBL6063814 0.82 CYP19A1 (0.38) CYP19A1CYP11B1CYP11B2
SCHEMBL8323116 0.82 CYP19A1 (0.39) CYP19A1KDM1ASTS
SCHEMBL27287580 0.81 CYP11B1 (0.44) CYP19A1CYP11B1CYP11B2STS
SCHEMBL8322680 0.80 CYP19A1 (0.45) CYP19A1STS
SCHEMBL8327702 0.80 CYP19A1 (0.36) CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113387894-A 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2021-09-14 CN claimed
CN-113387894-B 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2023-02-24 CN disclosed
CN-113387894-A 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2021-09-14 CN disclosed