SCHEMBL8327043

SCHEMBL8327043

N#Cc1ccc(N(Cc2ccc(F)c(F)c2)c2cncnc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 14/20 0.45
NR1D1 P20393 1/20 0.42
NR1H3 Q13133 1/20 0.42
STS P08842 2/20 0.39
CYP3A4 P08684 1/20 0.39
CTSL P07711 2/20 0.38
VNN1 O95497 1/20 0.37
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28922397 0.90 CYP19A1 (0.46) CYP19A1STSKDM1A
SCHEMBL8329384 0.89 CYP19A1 (0.43) CYP19A1NR1D1NR1H3STSCTSL
SCHEMBL8327987 0.89 CYP19A1 (0.42) CYP19A1STSCTSLVNN1
SCHEMBL8328066 0.86 CYP19A1 (0.44) CYP19A1STS
SCHEMBL8324262 0.86 CYP19A1 (0.40) CYP19A1STSCYP3A4VNN1
SCHEMBL8323103 0.85 ESR1 (0.49) CYP19A1NR1D1CTSLVNN1KDM1A
SCHEMBL6063814 0.84 CYP19A1 (0.38) CYP19A1CTSLVNN1
SCHEMBL8323116 0.84 CYP19A1 (0.39) CYP19A1STSCTSLVNN1KDM1A
SCHEMBL27287580 0.84 CYP11B1 (0.44) CYP19A1STSCTSL
SCHEMBL8329428 0.83 MAOA (0.42) CYP19A1NR1D1NR1H3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed