SCHEMBL8324327

SCHEMBL8324327

Nc1nc(O)c2c(n1)NC[C@H](CCc1ccc(Br)cc1)C2

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.47
GART P22102 3/20 0.41
NOS1 P29475 1/20 0.32
CHIT1 Q13231 2/20 0.31
CHIA Q9BZP6 2/20 0.31
COPS5 Q92905 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875735 1.00 DHFR (0.47) DHFRGARTNOS1CHIT1CHIA
SCHEMBL8326952 1.00 DHFR (0.47) DHFRGARTNOS1CHIT1CHIA
SCHEMBL8874134 0.86 DHFR (0.56) DHFRGARTNOS1
SCHEMBL7490675 0.86 DHFR (0.56) DHFRGARTNOS1
Hydrochloric Acid SCHEMBL8875657 0.85 DHFR (0.55) DHFRGARTNOS1
SCHEMBL9460931 0.85 DHFR (0.47) DHFRGARTNOS1CHIT1CHIA
Hydrochloric Acid SCHEMBL7487428 0.85 DHFR (0.55) DHFRGARTNOS1
SCHEMBL8875010 0.85 DHFR (0.45) DHFRGARTNOS1
SCHEMBL9709383 0.83 DHFR (0.43) DHFRGARTNOS1
SCHEMBL9460668 0.81 DHFR (0.41) DHFRGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593286-B1 Intermediates for preparing antifolate compounds and processes thereto LILLY CO ELI (US) 1999-12-15 EP disclosed
US-5981745-A μ-oxo-gallium phthalocyanine dimer having novel polymorph and electrophotographic photoreceptor prepared by using the same ORIENT CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-09 US disclosed
US-5969136-A Cyclization for preparing antifolate compounds ELI LILLY AND COMPANY (US) 1999-10-19 US disclosed
US-5910384-A FOR COPIERS, PRINTERS; PHOTOSENSITIVITY, DURABILITY ORIENT CHEMICAL INDUSTRIES, LTD. (JP) 1999-06-08 US disclosed
US-5486614-A Intermediates for preparing antifolate compounds ELI LILLY AND COMPANY (US) 1996-01-23 US disclosed
EP-0593286-A2 Intermediates for preparing antifolate compounds and processes there to ELI LILLY AND COMPANY (US) 1994-04-20 EP disclosed