SCHEMBL8875010

SCHEMBL8875010

N#Cc1ccc(CC[C@@H]2CNc3nc(N)nc(O)c3C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.45
GART P22102 3/20 0.39
HRH3 Q9Y5N1 1/20 0.38
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
NOS1 P29475 2/20 0.33
KCNJ1 P48048 1/20 0.32
KCNH2 Q12809 1/20 0.32
NOS3 P29474 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324327 0.85 DHFR (0.47) DHFRGARTNOS1
SCHEMBL7490675 0.83 DHFR (0.56) DHFRGARTNOS1
SCHEMBL8874134 0.83 DHFR (0.56) DHFRGARTNOS1
Hydrochloric Acid SCHEMBL7487428 0.83 DHFR (0.55) DHFRGARTNOS1
Hydrochloric Acid SCHEMBL8875657 0.83 DHFR (0.55) DHFRGARTNOS1
SCHEMBL9460931 0.83 DHFR (0.47) DHFRGARTMAOBNOS1NOS3
SCHEMBL9709383 0.80 DHFR (0.43) DHFRGARTNOS1KCNH2
SCHEMBL9460668 0.79 DHFR (0.41) DHFRGART
SCHEMBL9460927 0.78 DHFR (0.41) DHFRGARTMAOAMAOBNOS1
SCHEMBL9460872 0.76 MAOB (0.41) DHFRMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633373-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1997-05-27 US disclosed
EP-0407212-B1 Enantioselective synthesis of antifolates LILLY CO ELI (US) 1996-05-22 EP disclosed
US-5516776-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1996-05-14 US disclosed
US-5159090-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1992-10-27 US disclosed
US-5008391-A Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1991-04-16 US disclosed
EP-0407212-A1 Enantioselective synthesis of antifolates ELI LILLY AND COMPANY (US) 1991-01-09 EP disclosed