SCHEMBL8324645

SCHEMBL8324645

CC(C)(C)OC(=O)c1ccc(CCc2cncnc2Cl)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2C19 P33261 1/20 0.36
CKS1B P61024 1/20 0.36
SKP2 Q13309 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325834 0.80 NPC1 (0.43) ALDH1A1TP53HPGDALOX15HSD17B10
SCHEMBL8321963 0.76 CA12 (0.39) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL6260897 0.76 NAMPT (0.39) ALDH1A1TP53SIRT2SIRT1NAMPT
SCHEMBL8325953 0.74 PTGER1 (0.47) ALDH1A1HPGDRXRANR1H2HDAC1
SCHEMBL14966328 0.72 HDAC1 (0.50) ALDH1A1CYP1A2CYP2C19HSD17B10CA12
SCHEMBL4277492 0.71 ATR (0.40) ALDH1A1CSNK2A1KMT2A
SCHEMBL13891334 0.71 PLK1 (0.51) ALDH1A1CA12CA1CA2CA9
SCHEMBL2207588 0.71 CYP4A11 (0.60) ALDH1A1CYP2C9CYP2C19CA12CA1
SCHEMBL4212803 0.70 SIRT2 (0.43) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL7246822 0.70 CA12 (0.48) ALOX15CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed