SCHEMBL8321963

SCHEMBL8321963

CC(C)(C)OC(=O)c1ccc(CCc2cnc[nH]c2=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
HRH3 Q9Y5N1 4/20 0.37
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
CYP2C19 P33261 1/20 0.36
CKS1B P61024 1/20 0.36
SKP2 Q13309 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8320778 0.80 RARB (0.42) HRH3ALDH1A1TP53
SCHEMBL6260897 0.76 NAMPT (0.39) ALDH1A1TP53SIRT2SIRT1
SCHEMBL8324645 0.76 ALDH1A1 (0.36) CA12CA1CA2CA9CA14
SCHEMBL8325174 0.73 GABRA1 (0.45) CA12CA1CA2CA9CA14
SCHEMBL14966328 0.72 HDAC1 (0.50) CA12CA1CA2CA9CA14
SCHEMBL2207588 0.71 CYP4A11 (0.60) CA12CA1CA2CA9CA14
SCHEMBL13891334 0.71 PLK1 (0.51) CA12CA1CA2CA9CA14
SCHEMBL4212803 0.70 SIRT2 (0.43) CA12CA1CA2CA9CA14
SCHEMBL4057710 0.70 CA12 (0.55) CA12CA1CA2CA9CA14
SCHEMBL16594355 0.70 CA12 (0.50) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed