SCHEMBL8325834

SCHEMBL8325834

O=C(O)c1ccc(CCc2cncnc2Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TP53 P04637 1/20 0.43
HSD17B10 Q99714 1/20 0.41
NR4A2 P43354 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
NAPRT Q6XQN6 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TBXAS1 P24557 2/20 0.39
RARB P10826 2/20 0.39
HPGD P15428 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
MBOAT4 Q96T53 1/20 0.38
P2RX3 P56373 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324645 0.80 ALDH1A1 (0.36) RAB9ATP53HSD17B10ALDH1A1HPGD
Terephthalic Acid SCHEMBL4612225 0.73 TSHR (0.67) SMN1; SMN2TP53NAPRTALDH1A1RARB
SCHEMBL70166 0.73 TSHR (0.67) SMN1; SMN2TP53NAPRTALDH1A1RARB
SCHEMBL6257548 0.72 KDM6B (0.46) NPC1RAB9ASMN1; SMN2HSD17B10NAPRT
SCHEMBL16687966 0.71 ALDH1A1 (0.54) TP53ALDH1A1RARBP2RX3TSHR
SCHEMBL5751057 0.71 TSHR (0.74) NPC1RAB9ASMN1; SMN2TP53HSD17B10
Hydrochloric Acid SCHEMBL7132238 0.71 TSHR (0.63) TP53NAPRTALDH1A1RARBP2RX3
SCHEMBL907669 0.71 KDM4E (0.37) NFKB1NAPRTALDH1A1TSHRHCAR2
SCHEMBL8320778 0.71 RARB (0.42) NPC1RAB9ASMN1; SMN2TP53ALDH1A1
SCHEMBL6769826 0.70 NAPRT (0.64) NPC1RAB9ASMN1; SMN2TP53NAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed