SCHEMBL8324775

SCHEMBL8324775

O=C(O)/C=C/c1cccc(CC(=O)O)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.59
LTB4R2 Q9NPC1 1/20 0.59
KDM4E B2RXH2 5/20 0.59
ALDH1A1 P00352 3/20 0.59
PKM P14618 2/20 0.59
NPSR1 Q6W5P4 1/20 0.59
HDAC4 P56524 3/20 0.57
HDAC3 O15379 2/20 0.57
HDAC1 Q13547 2/20 0.57
HDAC7 Q8WUI4 2/20 0.57
HDAC2 Q92769 2/20 0.57
HDAC10 Q969S8 2/20 0.57
HDAC11 Q96DB2 2/20 0.57
HDAC8 Q9BY41 2/20 0.57
HDAC6 Q9UBN7 2/20 0.57
HDAC9 Q9UKV0 2/20 0.57
HDAC5 Q9UQL6 2/20 0.57
TNKS O95271 1/20 0.57
HCAR2 Q8TDS4 1/20 0.57
TNKS2 Q9H2K2 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10374325 1.00 LTB4R (0.59) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL4397023 0.91 AKR1B1 (0.56) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL4397024 0.91 AKR1B1 (0.56) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL3627668 0.86 LTB4R (0.60) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL3627671 0.86 LTB4R (0.60) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL18197880 0.86 AKR1B1 (0.50) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL2810112 0.84 TTR (0.51) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL2810114 0.84 TTR (0.51) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL30967860 0.84 TTR (0.51) LTB4RLTB4R2KDM4EALDH1A1PKM
SCHEMBL853486 0.84 NPSR1 (0.61) LTB4RLTB4R2KDM4EALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed
EP-0201823-B1 NOVEL INTERMEDIATES FOR THE PRODUCTION OF PHARMACEUTICALS LILLY INDUSTRIES LIMITED (GB) 1990-12-05 EP disclosed
US-4963578-A LEUKOTRIN ANTAGONISTS; ANTIALLERGENS LILLY INDUSTRIES LIMITED (GB) 1990-10-16 US disclosed
US-RE33300-E LEUKOTRIENE ANTAGONISTS; ANTIALLERGENS ELI LILLY AND COMPANY (US) 1990-08-14 US disclosed
EP-0134111-B1 ARALIPHATIC SULPHIDES,SULPHONES AND SULPHOXIDES AND THEIR PHARMACEUTICAL USE Lilly Industries Limited (GB) 1988-12-07 EP disclosed
US-4665189-A LEUKOTRIENE ANTAGONISTS LILLY INDUSTRIES LIMITED (GB) 1987-05-12 US disclosed
EP-0201823-A2 Novel intermediates for the production of pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1986-11-20 EP disclosed
EP-0134111-A1 Araliphatic sulphides,sulphones and sulphoxides and their pharmaceutical use Lilly Industries Limited (GB) 1985-03-13 EP disclosed