SCHEMBL8325158

SCHEMBL8325158

CC([CH]c1cccc2ccccc12)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.44
SIGMAR1 Q99720 4/20 0.44
SLC6A2 P23975 2/20 0.44
MAOA P21397 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP2A6 P11509 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
CAPN1 P07384 2/20 0.43
SMPD2 O60906 1/20 0.43
CTSB P07858 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.42
CTSL P07711 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4819774 0.81 SMPD2 (0.42) SMPD2ALDH1A1F2LMNA
SCHEMBL8322787 0.80 CAPN1 (0.49) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8325552 0.80 CAPN1 (0.41) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL6027641 0.79 SMPD2 (0.41) CYP2A6SMPD2ALDH1A1F2LMNA
SCHEMBL6707342 0.77 SMPD2 (0.43) SMPD2ALDH1A1CYP2D6F2LMNA
SCHEMBL3243723 0.76 ALDH1A1 (0.45) CYP2A6SMPD2ALDH1A1F2LMNA
SCHEMBL6709477 0.75 SMPD2 (0.39) SMPD2ALDH1A1MAPTF2LMNA
SCHEMBL7616489 0.74 SMPD2 (0.42) SLC6A4CYP2A6SMPD2ALDH1A1F2
SCHEMBL6709427 0.73 ALDH1A1 (0.50) SMPD2ALDH1A1F2LMNA
SCHEMBL4189468 0.70 ACP3 (0.55) TAAR1SIGMAR1SLC6A2MAOASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed