SCHEMBL8322787

SCHEMBL8322787

CNC([CH]c1cccc2ccccc12)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 2/20 0.49
CTSB P07858 1/20 0.43
TAAR1 Q96RJ0 4/20 0.42
SIGMAR1 Q99720 4/20 0.42
SLC18A2 Q05940 1/20 0.42
ACP3 P15309 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
CTSL P07711 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
SMPD2 O60906 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
MAOA P21397 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325158 0.80 TAAR1 (0.44) CAPN1CTSBTAAR1SIGMAR1SLC18A2
SCHEMBL8325552 0.76 CAPN1 (0.41) CAPN1CTSBTAAR1SIGMAR1ACP3
SCHEMBL8325444 0.70 TAAR1 (0.46) TAAR1SIGMAR1SLC18A2MEN1KMT2A
SCHEMBL8327429 0.70 TAAR1 (0.42) TAAR1SIGMAR1SLC18A2ALDH1A1POLB
SCHEMBL2920753 0.70 TAAR1 (0.53) CAPN1CTSBTAAR1SIGMAR1SLC18A2
SCHEMBL1970032 0.70 TAAR1 (0.53) CAPN1CTSBTAAR1SIGMAR1SLC18A2
SCHEMBL19559843 0.70 SIGMAR1 (0.53) TAAR1SIGMAR1SLC18A2MEN1KMT2A
SCHEMBL7607231 0.70 SIGMAR1 (0.53) TAAR1SIGMAR1SLC18A2MEN1KMT2A
SCHEMBL6852338 0.70 TAAR1 (0.53) CAPN1CTSBTAAR1SIGMAR1SLC18A2
SCHEMBL3243723 0.69 ALDH1A1 (0.45) ALDH1A1SMPD2MTNR1AMTNR1BCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed