SCHEMBL8325396

SCHEMBL8325396

COCc1nc(Cl)c(Oc2cc(OC)ccc2Cl)c(NS(=O)(=O)c2ccc3c(c2)OCO3)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
MAPT P10636 5/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 2/20 0.46
TSHR P16473 3/20 0.45
EDNRA P25101 2/20 0.45
USP2 O75604 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
LMNA P02545 2/20 0.41
GLA P06280 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.39
HTT P42858 1/20 0.39
SLC22A12 Q96S37 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
EDNRB P24530 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326435 0.92 EDNRA (0.45) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL9151761 0.88 ALDH1A1 (0.49) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL8324961 0.88 EDNRA (0.58) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL8324259 0.88 MAPT (0.46) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL7293555 0.84 MAPT (0.48) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL8325940 0.84 EDNRA (0.56) EDNRAEDNRB
SCHEMBL9154629 0.83 EDNRA (0.51) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL9152112 0.82 EDNRA (0.54) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL9152792 0.82 EDNRA (0.54) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL9157393 0.82 MAPT (0.45) ALDH1A1MAPTMEN1KMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633259-B1 Sulfonylaminopyrimidines, their preparation and their use as medicine HOFFMANN LA ROCHE (CH) 1999-01-13 EP disclosed
US-5541186-A ENDOTHELIN RECEPTOR INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1996-07-30 US disclosed
EP-0633259-A1 Sulfonylaminopyrimidines, their preparation and their use as medicine F. HOFFMANN-LA ROCHE AG (CH) 1995-01-11 EP disclosed