SCHEMBL8325558

SCHEMBL8325558

C=Cc1c(F)c(N2CC3C=CC=CC3(N)C2)cc2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.46
HRH3 Q9Y5N1 1/20 0.46
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 4/20 0.39
LMNA P02545 3/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPT P10636 1/20 0.39
TOP2A P11388 3/20 0.39
TOP2B Q02880 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 2/20 0.37
CACNA1F O60840 1/20 0.37
MAPK1 P28482 1/20 0.37
CACNA1D Q01668 1/20 0.37
CACNA1S Q13698 1/20 0.37
CACNA1C Q13936 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923870 0.95 KCNH2 (0.42) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL8325561 0.88 KCNH2 (0.34) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL8923882 0.87 KCNH2 (0.35) KCNH2HRH3ALDH1A1TOP2ATOP2B
SCHEMBL8323756 0.82 KDM4E (0.58) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8323773 0.78 MEN1 (0.60) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL8922496 0.77 MEN1 (0.58) KCNH2HRH3ALDH1A1TOP2ATOP2B
SCHEMBL8322412 0.77 CACNA1F (0.62) KCNH2TOP2ATOP2BMEN1KMT2A
SCHEMBL8322078 0.76 MEN1 (0.51) KCNH2HRH3ALDH1A1TOP2ATOP2B
SCHEMBL8322523 0.76 KMT2A (0.40) ALDH1A1KDM4ELMNAHPGDHSD17B10
SCHEMBL8324813 0.75 KCNH2 (0.53) KCNH2ALDH1A1KDM4ELMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705828-B1 Quinolone- and naphthyridone carboxylic acid derivatives as antibacterial agents BAYER AG (DE) 1999-12-01 EP disclosed
EP-0705828-A1 Quinolone- and naphthyridone carboxylic acid derivatives as antibacterial agents BAYER AG (DE) 1996-04-10 EP disclosed