SCHEMBL8923882

SCHEMBL8923882

C=Cc1c(F)c(N2CC3C=CC=CC3(N)C2)cc2c1c(=O)c(C(=O)OC(=O)c1cn(C3CC3)c3c(F)c(F)c(F)c(C=C)c3c1=O)cn2C1CC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.35
HRH3 Q9Y5N1 1/20 0.35
POLB P06746 2/20 0.32
CACNA1F O60840 1/20 0.32
MAPK1 P28482 1/20 0.32
CACNA1D Q01668 1/20 0.32
CACNA1S Q13698 1/20 0.32
CACNA1C Q13936 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
TOP2A P11388 1/20 0.30
TOP2B Q02880 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8923870 0.93 KCNH2 (0.42) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL8325558 0.87 KCNH2 (0.46) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL8325561 0.82 KCNH2 (0.34) KCNH2HRH3ALDH1A1TOP2ATOP2B
SCHEMBL8923856 0.78 KMT2A (0.33) POLBKMT2AALDH1A1
SCHEMBL8923183 0.75 KCNH2 (0.43) KCNH2POLBMEN1KMT2AALDH1A1
SCHEMBL8922496 0.73 MEN1 (0.58) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL8926299 0.73 ALDH1A1 (0.52) KCNH2POLBMEN1KMT2AALDH1A1
SCHEMBL8323773 0.71 MEN1 (0.60) KCNH2HRH3POLBCACNA1FMAPK1
SCHEMBL8323756 0.71 KDM4E (0.58) ALDH1A1TOP2ATOP2B
SCHEMBL8923852 0.70 KMT2A (0.39) POLBMEN1KMT2AALDH1A1TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679689-A BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-10-21 US disclosed