SCHEMBL8325630

SCHEMBL8325630

COC(=O)/C=C/c1ccc(Cn2cncc2C)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 8/20 0.48
CYP11B2 P19099 8/20 0.48
CYP19A1 P11511 1/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
TYR P14679 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
KDM4E B2RXH2 2/20 0.43
MAPT P10636 1/20 0.43
PTPN1 P18031 1/20 0.43
HDAC6 Q9UBN7 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319267 0.86 HDAC6 (0.55) CYP11B1CYP11B2CYP19A1HDAC6HDAC3
SCHEMBL7995117 0.85 CYP11B1 (0.52) CYP11B1CYP11B2CA12CA1CA2
SCHEMBL7995116 0.85 CYP11B1 (0.52) CYP11B1CYP11B2CA12CA1CA2
SCHEMBL21334813 0.77 CYP11B1 (0.56) CYP11B1CYP11B2CYP19A1HDAC6HDAC3
SCHEMBL9641646 0.76 CYP11B1 (0.54) CYP11B1CYP11B2KDM4EHDAC1HDAC8
SCHEMBL11107722 0.76 TBXAS1 (0.72) CYP11B1CYP11B2CYP19A1CYP1A2KMT2A
SCHEMBL11107726 0.76 TBXAS1 (0.72) CYP11B1CYP11B2CYP19A1CYP1A2KMT2A
SCHEMBL8324714 0.75 CA12 (0.48) CA12CA1CA2TYRCA7
SCHEMBL28052073 0.75 TBXAS1 (0.70) CYP11B1CYP11B2CYP19A1CYP1A2KMT2A
SCHEMBL8319380 0.74 HDAC6 (0.46) CYP11B1CYP11B2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed