SCHEMBL8325832

SCHEMBL8325832

Fc1ccc(-c2[c]c3ccccc3cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.39
CYP2A6 P11509 1/20 0.39
MAPK10 P53779 1/20 0.33
MAPK14 Q16539 1/20 0.33
CYP1A1 P04798 2/20 0.33
CYP1B1 Q16678 2/20 0.33
XDH P47989 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
KDM4E B2RXH2 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ADORA2A P29274 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.30
CYP3A4 P08684 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3149589 0.84 ALDH1A1 (0.38) CYP1A2CYP1A1CYP1B1CYP3A4
SCHEMBL79020 0.84 ALDH1A1 (0.35) CYP2A6RAB9AMEN1KMT2A
SCHEMBL28957329 0.81 CYP1A2 (0.41) CYP1A2CYP2A6CYP1A1CYP1B1NPC1
SCHEMBL8359885 0.81 MEN1 (0.42) CYP1A2NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL321122 0.81 TDP1 (0.39) CYP1A2CYP2A6NPC1RAB9AKDM4E
SCHEMBL7139286 0.81 ALDH1A1 (0.41) CYP1A2CYP2A6MAPK14CYP1A1CYP1B1
SCHEMBL9418157 0.81 ESR1 (0.47) CYP1A2NPC1RAB9AHPGDMEN1
SCHEMBL5785358 0.80 KIF11 (0.47) MAPK14
SCHEMBL239122 0.79 CYP2A6 (0.37) CYP1A2CYP2A6CYP1A1CYP1B1CYP3A4
SCHEMBL1719526 0.78 GSTP1 (0.44) CYP1A2CYP1A1CYP1B1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed
US-4455421-A ANTIFERTILITY, ANTIULCER AGENTS; TETRAZOLE DERIVATIVES PFIZER INC. (US) 1984-06-19 US disclosed
US-4365077-A ANTIFERTILITY, ANTIULCER PFIZER INC. (US) 1982-12-21 US disclosed
US-4157341-A 11-Desoxy-16-aryloxy-ω-tetranorprostaglandins PFIZER INC. (US) 1979-06-05 US disclosed