SCHEMBL8325934

SCHEMBL8325934

CC(C)(C)OC(=O)N[C@@H]1C[C@@]12CCc1cc3ccccc3n1C2

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
EPHX2 P34913 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
NR1H2 P55055 6/20 0.34
PPIA P62937 1/20 0.34
DRD2 P14416 2/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
CKS1B P61024 1/20 0.33
SKP1 P63208 1/20 0.33
SKP2 Q13309 1/20 0.33
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
KDM4A O75164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327513 1.00 HTR2A (0.34) HTR2AHTR2CEPHX2SIGMAR1NR1H2
SCHEMBL8653934 0.75 KMT2A (0.46) EPHX2SIGMAR1DRD2KMT2AL3MBTL1
SCHEMBL8328030 0.73 HTR2A (0.39) HTR2AHTR2CSIGMAR1
SCHEMBL6590757 0.72 KCNA3 (0.50) EPHX2SIGMAR1DRD2KMT2AL3MBTL1
SCHEMBL8329435 0.72 HTR2A (0.39) HTR2AHTR2CKMT2A
SCHEMBL8322785 0.71 HTR2A (0.47) HTR2AHTR2CSIGMAR1KDM1AMAOB
SCHEMBL8328872 0.71 HTR2A (0.47) HTR2AHTR2CSIGMAR1KDM1AMAOB
SCHEMBL21028327 0.71 HTR2A (0.42) HTR2AHTR2CSIGMAR1KMT2A
SCHEMBL8322544 0.67 HTR2A (0.40) HTR2AHTR2CSIGMAR1
SCHEMBL6947042 0.67 PDE4B (0.44) KMT2AL3MBTL1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed