SCHEMBL8329435

SCHEMBL8329435

CCOC(=O)C1CC12CCc1cc3ccccc3n1C2

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.39
HTR2C P28335 4/20 0.39
NOD2 Q9HC29 5/20 0.36
NOD1 Q9Y239 5/20 0.36
OPRM1 P35372 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 2/20 0.34
TSHR P16473 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328030 0.83 HTR2A (0.39) HTR2AHTR2COPRM1
SCHEMBL8320925 0.76 HTR2A (0.42) HTR2AHTR2COPRM1MEN1KMT2A
SCHEMBL8328343 0.74 ALDH1A1 (0.45) HTR2AHTR2CKDM4EALDH1A1
SCHEMBL8322785 0.73 HTR2A (0.47) HTR2AHTR2C
SCHEMBL8328872 0.73 HTR2A (0.47) HTR2AHTR2C
SCHEMBL8657721 0.73 ALDH1A1 (0.49) HTR2AHTR2CMEN1KMT2APKM
SCHEMBL8325934 0.72 HTR2A (0.34) HTR2AHTR2CKMT2A
SCHEMBL8447552 0.71 ALDH1A1 (0.44) MEN1KMT2APKMRAB9AKDM4E
SCHEMBL21028327 0.71 HTR2A (0.42) HTR2AHTR2CMEN1KMT2A
SCHEMBL3156042 0.69 HTR2A (0.46) HTR2AHTR2COPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed