SCHEMBL8326415

SCHEMBL8326415

Cc1c(CCO)[nH]c2ncccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.40
AURKA O14965 1/20 0.40
PARP1 P09874 1/20 0.40
FEN1 P39748 1/20 0.40
NPC1 O15118 1/20 0.39
HSP90AA1 P07900 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PDK2 Q15119 2/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
MTNR1A P48039 1/20 0.37
GPR84 Q9NQS5 1/20 0.37
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
RET P07949 1/20 0.36
CCNB1 P14635 1/20 0.36
CCNB3 Q8WWL7 1/20 0.36
KIT P10721 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328576 0.87 AURKA (0.42) RIPK1AURKAPARP1FEN1NPC1
SCHEMBL9386690 0.81 KDM4E (0.40) RIPK1AURKAPARP1FEN1NPC1
SCHEMBL8329539 0.77 PKM (0.43) AURKAPARP1FEN1NPC1HSP90AA1
SCHEMBL30324482 0.73 KDM4E (0.50) AURKAPARP1FEN1NPC1HSP90AA1
SCHEMBL855363 0.73 KDM4E (0.50) AURKAPARP1FEN1NPC1HSP90AA1
SCHEMBL31405650 0.73 ALDH1A1 (0.59) ALDH1A1TSHRHTTKMT2AMAPT
SCHEMBL3921386 0.71 HTT (0.39) RIPK1AURKAPARP1FEN1ALDH1A1
SCHEMBL21115235 0.70 AURKA (0.46) AURKAPARP1FEN1NPC1HSP90AA1
SCHEMBL8324581 0.70 AURKA (0.46) AURKAPARP1FEN1NPC1HSP90AA1
SCHEMBL28329874 0.70 AXL (0.47) AURKAPARP1FEN1NPC1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509974-B1 Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof ASTRA AB (SE) 1999-01-13 EP disclosed
EP-0509974-A1 Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof Astra Aktiebolag (SE) 1992-10-21 EP disclosed