SCHEMBL8326729

SCHEMBL8326729

CCOC(=S)C(C)(C(=O)O)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TDP1 Q9NUW8 2/20 0.43
CYP3A4 P08684 2/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
KCNA5 P22460 1/20 0.41
RORC P51449 1/20 0.40
CDC7 O00311 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 3/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MAPT P10636 2/20 0.38
CYP17A1 P05093 2/20 0.38
CYP19A1 P11511 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326723 0.89 KCNA5 (0.43) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL3949682 0.86 MAPK1 (0.46) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL8330075 0.81 MAPK1 (0.49) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL10772486 0.81 LMNA (0.57) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL8326726 0.80 MAPK1 (0.45) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL1225868 0.76 TDP1 (0.56) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL1605423 0.74 MAPK1 (0.48) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL8326720 0.74 MAPK1 (0.43) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL9394785 0.73 MAPK1 (0.47) ALDH1A1TDP1CYP3A4LMNACYP1A2
SCHEMBL8330071 0.73 SMN1; SMN2 (0.44) ALDH1A1TDP1CYP3A4LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908863-A ANTIGROWTH AGENT FOR BONES DOMPE' S.P.A. (IT) 1999-06-01 US disclosed
EP-0792878-A2 Geminal carboxylic acids and esters thereof, pharmaceutical formulations containing them useful in the treatment of bone dysmetabolism Dompé S.P.A. (IT) 1997-09-03 EP disclosed