SCHEMBL8327006

SCHEMBL8327006

[CH2]C(C)C(c1ccccc1)c1ccc(F)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.48
SLC6A4 P31645 3/20 0.48
SLC6A3 Q01959 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
KCNH2 Q12809 1/20 0.48
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TSHR P16473 2/20 0.36
KDM4E B2RXH2 1/20 0.36
PTGS2 P35354 1/20 0.36
SOS1 Q07889 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
PLA2G1B P04054 1/20 0.36
CYP1A2 P05177 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327275 0.83 SLC6A4 (0.51) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8319057 0.80 ACP3 (0.45) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL16958488 0.77 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8326598 0.77 NPC1 (0.42) SLC6A4CYP3A4CYP2D6NPC1KDM4E
SCHEMBL2093738 0.76 MIF (0.43) CYP2D6TSHRKDM4ELMNAALDH1A1
SCHEMBL8330722 0.76 IDO1 (0.46) SLC6A2SLC6A4KDM4EIDO1TDO2
SCHEMBL8326192 0.73 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL530400 0.73 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL17486766 0.73 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL16951405 0.73 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed