SCHEMBL8330722

SCHEMBL8330722

[CH2]C(C)C(c1ccccc1)c1cccc(F)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
MTOR P42345 1/20 0.41
SLC6A4 P31645 3/20 0.39
SLC6A2 P23975 2/20 0.39
CNR2 P34972 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
KDM4E B2RXH2 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ACHE P22303 1/20 0.38
AOC3 Q16853 1/20 0.37
NFE2L2 Q16236 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL683672 0.85 IDO1 (0.49) IDO1TDO2MTORSLC6A4SLC6A2
SCHEMBL8326598 0.82 NPC1 (0.42) SLC6A4KDM4E
SCHEMBL2093738 0.82 MIF (0.43) KDM4E
SCHEMBL8324360 0.81 HDAC4 (0.40) HDAC4KDM4E
SCHEMBL8325753 0.81 AOC3 (0.44) IDO1TDO2MTORSLC6A4SLC6A2
SCHEMBL8328722 0.81 IDO1 (0.42) IDO1TDO2MTORSLC6A4SLC6A2
SCHEMBL8324324 0.79 ACP3 (0.46) ACHEAOC3OPRM1OPRD1OPRK1
SCHEMBL28597604 0.78 ACHE (0.44) IDO1TDO2MTORSLC6A4SLC6A2
SCHEMBL10442326 0.78 AOC3 (0.46) IDO1TDO2MTORSLC6A4HDAC4
SCHEMBL8323859 0.78 MAOA (0.41) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed