SCHEMBL8326192

SCHEMBL8326192

[CH2]CC(c1ccccc1)c1ccc(F)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.50
SLC6A4 P31645 4/20 0.50
CYP2D6 P10635 3/20 0.50
SLC6A3 Q01959 3/20 0.50
CYP3A4 P08684 2/20 0.50
KCNH2 Q12809 1/20 0.50
PLA2G1B P04054 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SOS1 Q07889 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
IDO2 Q6ZQW0 1/20 0.36
HTT P42858 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7429108 0.79 IDO1 (0.50) SLC6A2SLC6A4CYP2D6SLC6A3KCNH2
SCHEMBL8324166 0.78 ACP3 (0.47) SLC6A2SLC6A4IDO1TDO2HTT
SCHEMBL7430169 0.75 CYP19A1 (0.44) SLC6A4CYP2D6CYP3A4CYP1A2CYP2C9
SCHEMBL8325499 0.74 IDO1 (0.49) SLC6A2SLC6A4IDO1TDO2
SCHEMBL13126260 0.74 SLC6A2 (0.48) SLC6A2SLC6A4CYP2D6SLC6A3CYP3A4
SCHEMBL94275 0.74 HTR2A (0.52) RAB9ATDP1TSHR
SCHEMBL8327006 0.73 SLC6A2 (0.48) SLC6A2SLC6A4CYP2D6SLC6A3CYP3A4
SCHEMBL16950377 0.73 SLC6A2 (0.47) SLC6A2SLC6A4CYP2D6SLC6A3CYP3A4
SCHEMBL16960998 0.73 SLC6A2 (0.43) SLC6A2SLC6A4CYP2D6SLC6A3CYP3A4
SCHEMBL4635178 0.72 TSHR (0.44) SLC6A4CYP2D6SLC6A3CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed