SCHEMBL8327237

SCHEMBL8327237

COC(=O)c1ccc(/C=C/c2ccccc2OCc2ccccc2)c(Br)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
POLB P06746 1/20 0.55
PKM P14618 1/20 0.55
BLM P54132 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
PTGER1 P34995 1/20 0.54
PTGER4 P35408 1/20 0.54
PTGER3 P43115 1/20 0.54
PTGER2 P43116 1/20 0.54
LMNA P02545 5/20 0.51
MAPT P10636 3/20 0.51
GAA P10253 2/20 0.51
RAB9A P51151 2/20 0.51
ALDH1A1 P00352 2/20 0.51
NPC1 O15118 1/20 0.51
HPGD P15428 2/20 0.49
CCNB2 O95067 1/20 0.49
CDK1 P06493 1/20 0.49
CDK4 P11802 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8680186 1.00 MEN1 (0.55) MEN1KMT2APOLBPKMBLM
SCHEMBL8327239 1.00 MEN1 (0.55) MEN1KMT2APOLBPKMBLM
SCHEMBL8323954 0.89 PTGER1 (0.54) MEN1KMT2APOLBPKMBLM
SCHEMBL8323956 0.89 PTGER1 (0.54) MEN1KMT2APOLBPKMBLM
SCHEMBL8323795 0.88 MEN1 (0.57) MEN1KMT2APOLBPKMBLM
SCHEMBL8323794 0.88 MEN1 (0.57) MEN1KMT2APOLBPKMBLM
SCHEMBL8319292 0.88 PTGER1 (0.59) MEN1KMT2APTGER1PTGER4PTGER3
SCHEMBL8319297 0.88 PTGER1 (0.59) MEN1KMT2APTGER1PTGER4PTGER3
SCHEMBL8321308 0.87 LMNA (0.60) MEN1KMT2APOLBPKMBLM
SCHEMBL8321304 0.87 LMNA (0.60) MEN1KMT2APOLBPKMBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed