SCHEMBL8327670

SCHEMBL8327670

CC(=O)OC[C@H]1O[C@@H](n2cc(F)c(=O)[nH]c2=O)C[C@@H]1OCc1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TYMS P04818 1/20 0.44
RNASE1 P07998 1/20 0.40
TK2 O00142 2/20 0.39
TK1 P04183 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327674 1.00 LMNA (0.48) LMNASMN1; SMN2TYMSRNASE1TK2
SCHEMBL9098312 0.91 TYMS (0.53) LMNASMN1; SMN2TYMSRNASE1TK1
SCHEMBL9098319 0.91 TYMS (0.53) LMNASMN1; SMN2TYMSRNASE1TK1
SCHEMBL9339215 0.90 LMNA (0.46) LMNASMN1; SMN2TYMSRNASE1TK2
SCHEMBL8323429 0.90 TYMS (0.47) LMNASMN1; SMN2TYMSRNASE1TK1
SCHEMBL8323433 0.90 TYMS (0.47) LMNASMN1; SMN2TYMSRNASE1TK1
SCHEMBL8328242 0.89 LMNA (0.46) LMNASMN1; SMN2TYMSRNASE1TK1
Hydrochloric Acid SCHEMBL9339114 0.89 LMNA (0.46) LMNASMN1; SMN2TYMSRNASE1TK2
SCHEMBL8328237 0.89 LMNA (0.46) LMNASMN1; SMN2TYMSRNASE1TK1
Hydrochloric Acid SCHEMBL9339117 0.89 LMNA (0.46) LMNASMN1; SMN2TYMSRNASE1TK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0323441-B1 5-Fluorouracil derivatives OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP claimed
US-5869464-A HAVING LOW TOXICITY, SUSTAINING LOW CONCENTRATION IN BLOOD FOR EXTENDED PERIOD TAIHO PHARMACEUTICAL CO. LTD. (JP) 1999-02-09 US disclosed
EP-0686641-B1 2'-DEOXY-5-FLUOROURIDINE DERIVATIVE, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR DRUG TAIHO PHARMACEUTICAL CO LTD (JP) 1998-08-26 EP disclosed
EP-0323441-B1 5-Fluorouracil derivatives OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
EP-0686641-A1 2'-DEOXY-5-FLUOROURIDINE DERIVATIVE, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR DRUG TAIHO PHARMACEUTICAL CO., LTD. (JP) 1995-12-13 EP disclosed
US-5155113-A Administering 5-fluorouracil and derivatives with pyridine and pyridone derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-10-13 US disclosed
EP-0180188-B1 A COMPOSITION FOR INCREASING THE ANTI-CANCER ACTIVITY OF AN ANTI-CANCER COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-04-15 EP disclosed
US-4983609-A Anticancer agents OTSUKA PHARMACEUTICAL (JP) 1991-01-08 US disclosed
US-4864021-A ANTICARCINOGENIC AGENTS, ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-09-05 US disclosed
EP-0323441-A2 5-Fluorouracil derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-07-05 EP disclosed
EP-0180897-A2 5-Fluorouracil derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-05-14 EP disclosed
EP-0180188-A2 A composition for increasing the anti-cancer activity of an anti-cancer compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-05-07 EP disclosed