SCHEMBL8328131

SCHEMBL8328131

ClC1(Cl)CCn2c(ccc2-c2cccnc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
HK1 P19367 1/20 0.41
HKDC1 Q2TB90 1/20 0.41
CYP2D6 P10635 1/20 0.41
HIF1A Q16665 1/20 0.41
CYP2A6 P11509 6/20 0.38
ALDH1A1 P00352 4/20 0.38
CYP2A13 Q16696 1/20 0.38
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
DYRK3 O43781 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327314 0.74 CYP11B2 (0.37) CYP1A2HSD17B10CYP2A6ALDH1A1CYP2A13
SCHEMBL7856161 0.74 CHRNB4 (0.44) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL8328584 0.72 MKNK1 (0.44) CYP11B2
SCHEMBL8028928 0.71 CYP1A2 (0.47) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL929352 0.71 MKNK1 (0.43) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL10738674 0.69 CYP2A6 (0.44) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL2752518 0.69 MKNK1 (0.40) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL2344003 0.64 CYP11B1 (0.36) CYP1A2CYP3A4CYP2A6ALDH1A1LMNA
SCHEMBL6951232 0.64 CYP2A6 (0.61) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19
SCHEMBL8331912 0.64 CYP2A6 (0.41) CYP1A2CYP3A4HSD17B10CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946555-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 1999-10-06 EP claimed
WO-1998025925-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1998-06-18 WO claimed