SCHEMBL8328185

SCHEMBL8328185

CCOC(=O)c1ccc(/C=C\Cc2ccc(NC(C)=O)cc2OCc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPIA P62937 2/20 0.49
RAB9A P51151 4/20 0.47
KMT2A Q03164 4/20 0.46
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 3/20 0.46
CYP19A1 P11511 1/20 0.46
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
MAPT P10636 2/20 0.44
NAMPT P43490 1/20 0.44
GAA P10253 2/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
BRD4 O60885 2/20 0.43
NPC1 O15118 2/20 0.43
PTGER4 P35408 1/20 0.42
PTGER3 P43115 1/20 0.42
PTGER2 P43116 1/20 0.42
ALDH1A1 P00352 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328187 1.00 PPIA (0.49) PPIARAB9AKMT2AKDM4EMEN1
SCHEMBL8322219 0.82 PTGER1 (0.52) PPIARAB9AKMT2AKDM4EMEN1
SCHEMBL8322247 0.77 CYP19A1 (0.56) PPIARAB9AKMT2AKDM4EMEN1
SCHEMBL8677127 0.76 RAB9A (0.56) PPIARAB9AKMT2AKDM4EMEN1
SCHEMBL8327466 0.72 PTGER1 (0.54) KMT2AKDM4EMAPTPTGER4PTGER3
SCHEMBL8322906 0.72 PTGER4 (0.47) KDM4EPTGER4PTGER3PTGER2ALDH1A1
SCHEMBL8327463 0.72 PTGER1 (0.54) KMT2AKDM4EMAPTPTGER4PTGER3
SCHEMBL8322908 0.72 PTGER4 (0.47) KDM4EPTGER4PTGER3PTGER2ALDH1A1
SCHEMBL8459732 0.71 PTGER1 (0.66) RAB9AKMT2AKDM4EMEN1CYP19A1
SCHEMBL20691188 0.70 KMT2A (0.74) RAB9AKMT2AKDM4EMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed