SCHEMBL8328659

SCHEMBL8328659

Cc1c(C(=O)O)c2n(c1-c1cccnc1)CCC=C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.38
MKNK1 Q9BUB5 2/20 0.38
MKNK2 Q9HBH9 2/20 0.38
TBXAS1 P24557 2/20 0.38
KMO O15229 2/20 0.36
CYP11B2 P19099 2/20 0.36
DHODH Q02127 2/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
CYP2A6 P11509 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2E1 P05181 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP11B1 P15538 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963271 0.91 CYP2A6 (0.38) GPR35MKNK1MKNK2TBXAS1CYP11B2
SCHEMBL7965530 0.90 MKNK1 (0.40) MKNK1MKNK2TBXAS1CYP11B2LMNA
SCHEMBL7963752 0.88 SLC2A1 (0.39) CYP11B2LMNACYP3A4CYP11B1ALDH1A1
SCHEMBL8328721 0.86 MKNK1 (0.38) MKNK1MKNK2KMOCYP11B2CYP2A6
SCHEMBL8327786 0.85 CYP11B2 (0.37) MKNK1MKNK2KMOCYP11B2HTT
SCHEMBL8329319 0.84 CYP11B2 (0.38) MKNK1MKNK2KMOCYP11B2KDM4E
SCHEMBL8327305 0.83 MKNK1 (0.36) MKNK1MKNK2KMOCYP11B2CYP2C9
SCHEMBL7963276 0.81 CYP11B2 (0.39) MKNK1MKNK2CYP11B2KDM4ECYP2A6
SCHEMBL7962951 0.79 CYP11B2 (0.37) MKNK1MKNK2CYP11B2HTTCYP2A6
SCHEMBL7961877 0.79 CYP11B2 (0.40) CYP11B2KDM4EHTTCYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946555-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Aventis Pharma S.A. (FR) 1999-10-06 EP disclosed
WO-1998025925-A1 PYRROLE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM RHONE-POULENC RORER S.A. (FR) 1998-06-18 WO disclosed