SCHEMBL8329118

SCHEMBL8329118

O=C1Nc2c(ccc3c2CCNC3)/C1=N/O

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CD44 P16070 2/20 0.36
PARP1 P09874 2/20 0.32
TNKS2 Q9H2K2 1/20 0.32
PARP2 Q9UGN5 1/20 0.32
ACHE P22303 1/20 0.31
PNMT P11086 3/20 0.31
MAOB P27338 1/20 0.31
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329120 1.00 CD44 (0.36) CD44PARP1TNKS2PARP2ACHE
SCHEMBL8327813 0.81 CES1 (0.41) CD44PARP1TNKS2PARP2PNMT
SCHEMBL8328386 0.79 CA12 (0.30)
SCHEMBL8325695 0.75 MAOA (0.34) MAOB
SCHEMBL8325697 0.75 MAOA (0.34) MAOB
SCHEMBL3842153 0.75 PRCP (0.40)
SCHEMBL8330434 0.74 PARP1 (0.33) PARP1
SCHEMBL8330432 0.74 PARP1 (0.33) PARP1
SCHEMBL8329608 0.74
SCHEMBL8328966 0.72 ALDH1A1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed