SCHEMBL8329351

SCHEMBL8329351

CCCC(=O)N(C)C1CC1c1cccc(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
HTR2B P41595 2/20 0.47
SLC9A1 P19634 1/20 0.46
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
MTNR1B P49286 2/20 0.41
MTNR1A P48039 1/20 0.41
DRD2 P14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8332882 1.00 HTR2A (0.47) HTR2AHTR2CHTR2BSLC9A1CHRM2
SCHEMBL8333441 0.92 SLC9A1 (0.39) HTR2AHTR2CHTR2BSLC9A1CHRM2
SCHEMBL8333438 0.92 SLC9A1 (0.39) HTR2AHTR2CHTR2BSLC9A1CHRM2
SCHEMBL8330683 0.90 HTR2A (0.49) HTR2AHTR2CHTR2BSLC9A1CHRM2
SCHEMBL8331305 0.87 HTR2A (0.46) HTR2AHTR2CHTR2BSLC9A1CHRM2
SCHEMBL8332123 0.86 HTR2A (0.48) HTR2AHTR2CHTR2BSLC9A1CHRM2
SCHEMBL8331359 0.84 HTR2A (0.43) HTR2AHTR2CHTR2BDRD2
SCHEMBL8331482 0.84 HTR2C (0.43) HTR2AHTR2CHTR2BDRD2
SCHEMBL8331603 0.84 HTR2A (0.43) HTR2AHTR2CHTR2BDRD2
SCHEMBL8332789 0.83 SLC9A1 (0.51) HTR2AHTR2CHTR2BSLC9A1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US claimed
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed