SCHEMBL8333441

SCHEMBL8333441

[2H]C([2H])([2H])Oc1cccc(C2CC2N(C)C(=O)CCC)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
SIGMAR1 Q99720 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
ALOX5 P09917 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
GPR88 Q9GZN0 1/20 0.35
KDM1A O60341 1/20 0.34
RCOR1 Q9UKL0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8333438 1.00 SLC9A1 (0.39) SLC9A1HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8329351 0.92 HTR2A (0.47) SLC9A1HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8332882 0.92 HTR2A (0.47) SLC9A1HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8330683 0.82 HTR2A (0.49) SLC9A1HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8331603 0.81 HTR2A (0.43) HTR2AHTR2CHTR2BSLC6A4GPR88
SCHEMBL8331359 0.81 HTR2A (0.43) HTR2AHTR2CHTR2BKDM1A
SCHEMBL8331482 0.81 HTR2C (0.43) HTR2AHTR2CHTR2BGPR88
SCHEMBL8332792 0.80 HTR2A (0.43) SLC9A1HTR2AHTR2CHTR2B
SCHEMBL8469011 0.80 SLC5A1 (0.41) SIGMAR1
SCHEMBL8469013 0.80 SLC5A1 (0.41) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed