SCHEMBL8329359

SCHEMBL8329359

O=C1Nc2c(ccc3c2COC3)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 8/20 0.43
DAO P14920 2/20 0.40
NSD2 O96028 1/20 0.40
BCHE P06276 1/20 0.40
LIG1 P18858 1/20 0.37
PARP1 P09874 1/20 0.37
CASP3 P42574 1/20 0.33
CASP2 P42575 1/20 0.33
CASP7 P55210 1/20 0.33
CASP6 P55212 1/20 0.33
CASP8 Q14790 1/20 0.33
TGM2 P21980 2/20 0.33
DNMT1 P26358 1/20 0.33
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ALDH2 P05091 1/20 0.31
ALDH3A1 P30838 1/20 0.31
TDP2 O95551 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330434 0.80 PARP1 (0.33) PARP1
SCHEMBL8330432 0.80 PARP1 (0.33) PARP1
SCHEMBL2251074 0.77 PARP1 (0.57) CES1DAONSD2BCHELIG1
SCHEMBL2254584 0.74 PARP1 (0.53) CES1DAONSD2BCHELIG1
SCHEMBL8330690 0.74 CES1 (0.44) CES1DAONSD2BCHELIG1
SCHEMBL8330728 0.72 CES1 (0.43) CES1DAONSD2BCHELIG1
SCHEMBL8329643 0.71 CES1 (0.42) CES1DAONSD2BCHELIG1
SCHEMBL8327753 0.70 CES1 (0.42) CES1DAONSD2BCHELIG1
SCHEMBL8327813 0.70 CES1 (0.41) CES1DAONSD2BCHELIG1
SCHEMBL4391519 0.70 PNMT (0.44) CES1DAONSD2BCHELIG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116925100-A Substituted thiophenoquinolinone compound and preparation method and application thereof 深圳信立泰药业股份有限公司 2023-10-24 CN disclosed
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed