SCHEMBL8327753

SCHEMBL8327753

CN1Cc2ccc3c(c2C1)NC(=O)C3=O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.42
DAO P14920 2/20 0.41
NSD2 O96028 1/20 0.38
BCHE P06276 1/20 0.38
LIG1 P18858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 2/20 0.33
ALDH2 P05091 1/20 0.33
ALDH3A1 P30838 1/20 0.33
PARP1 P09874 1/20 0.32
CASP3 P42574 1/20 0.32
CASP2 P42575 1/20 0.32
CASP7 P55210 1/20 0.32
CASP6 P55212 1/20 0.32
CASP8 Q14790 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326465 0.86 CES1 (0.40) CES1DAONSD2BCHEL3MBTL1
SCHEMBL8328965 0.81 ALDH1A1 (0.30) ALDH1A1
SCHEMBL8328966 0.81 ALDH1A1 (0.30) ALDH1A1
SCHEMBL8329206 0.80 CES1 (0.40) CES1DAONSD2BCHELIG1
SCHEMBL8331316 0.80 CES1 (0.40) CES1DAONSD2BCHELIG1
SCHEMBL8331051 0.80 CES1 (0.40) CES1DAONSD2BCHELIG1
SCHEMBL8331553 0.73 ALDH1A1 (0.49) CES1DAONSD2BCHEALDH1A1
SCHEMBL8329239 0.73 CES1 (0.47) CES1DAONSD2BCHEL3MBTL1
SCHEMBL8330647 0.73 BCHE (0.43) CES1DAONSD2BCHEALDH1A1
SCHEMBL2257179 0.73 NOTUM (0.46) CES1LIG1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed