SCHEMBL8329372

SCHEMBL8329372

O=C(Cc1cccnc1)Nc1ccc(CCCc2ccccc2OCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.57
DRD2 P14416 2/20 0.57
PTGER1 P34995 2/20 0.56
PTGER4 P35408 1/20 0.56
PTGER3 P43115 1/20 0.56
PTGER2 P43116 1/20 0.56
ADRB1 P08588 3/20 0.50
ADRB3 P13945 3/20 0.50
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
SGMS2 Q8NHU3 1/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TRPV1 Q8NER1 1/20 0.48
IDO1 P14902 1/20 0.48
RAB9A P51151 1/20 0.47
ABCB1 P08183 1/20 0.47
CHRNA7 P36544 1/20 0.47
ADRB2 P07550 1/20 0.46
CYP11B1 P15538 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8676947 0.90 HTR1A (0.54) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8327887 0.89 PTGER1 (0.49) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8319651 0.88 CYP11B1 (0.57) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8676954 0.88 HTR1A (0.56) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8322148 0.85 PTGER1 (0.48) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8323432 0.85 PTGER1 (0.57) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8327698 0.81 PTGER1 (0.78) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8322518 0.81 PTGER1 (0.63) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8327425 0.79 PTGER1 (0.61) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8325504 0.78 HTR1A (0.60) HTR1ADRD2PTGER1PTGER4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed