SCHEMBL8322148

SCHEMBL8322148

CC(C)(O)C(=O)Nc1ccc(OCc2ccccc2)c(CCCc2ccc(NC(=O)Cc3cccnc3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 2/20 0.48
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
ADRB1 P08588 2/20 0.43
ADRB3 P13945 2/20 0.43
ITGB1 P05556 3/20 0.43
ITGA4 P13612 3/20 0.43
TRPV1 Q8NER1 1/20 0.43
P2RX4 Q99571 1/20 0.43
LRRK2 Q5S007 6/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PTGER4 P35408 1/20 0.41
PTGER3 P43115 1/20 0.41
PTGER2 P43116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319651 0.90 CYP11B1 (0.57) PTGER1CYP11B1CYP11B2HTR1ADRD2
SCHEMBL8327887 0.85 PTGER1 (0.49) PTGER1CYP11B1CYP11B2HTR1ADRD2
SCHEMBL8329372 0.85 HTR1A (0.57) PTGER1CYP11B1CYP11B2HTR1ADRD2
SCHEMBL8676947 0.80 HTR1A (0.54) PTGER1CYP11B1CYP11B2HTR1ADRD2
SCHEMBL8676954 0.74 HTR1A (0.56) PTGER1HTR1ADRD2LRRK2MEN1
SCHEMBL8324167 0.72 PTGER1 (0.51) PTGER1MEN1KMT2APTGER4PTGER3
SCHEMBL8323432 0.71 PTGER1 (0.57) PTGER1HTR1ADRD2ADRB1ADRB3
SCHEMBL8320635 0.69 MEN1 (0.56) PTGER1CYP11B1CYP11B2MEN1KMT2A
SCHEMBL9058743 0.69 PTGER1 (0.69) PTGER1MEN1KMT2APTGER4PTGER3
SCHEMBL8319393 0.68 PTGER1 (0.61) PTGER1HTR1ADRD2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed