SCHEMBL8329384

SCHEMBL8329384

N#Cc1ccc(N(Cc2ccc(Br)c(F)c2)c2cncnc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 16/20 0.43
STS P08842 3/20 0.37
CTSL P07711 1/20 0.36
NR1D1 P20393 1/20 0.35
NR1H3 Q13133 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327987 0.91 CYP19A1 (0.42) CYP19A1STSCTSLCYP11B1CYP11B2
SCHEMBL8327043 0.89 CYP19A1 (0.45) CYP19A1STSCTSLNR1D1NR1H3
SCHEMBL28922397 0.87 CYP19A1 (0.46) CYP19A1STSCYP11B1CYP11B2
SCHEMBL8328066 0.83 CYP19A1 (0.44) CYP19A1STSCYP11B1CYP11B2
SCHEMBL8325528 0.82 CYP19A1 (0.53) CYP19A1CYP11B1CYP11B2
SCHEMBL8323103 0.82 ESR1 (0.49) CYP19A1CTSLNR1D1CYP11B1CYP11B2
SCHEMBL30262479 0.82 CYP19A1 (0.41) CYP19A1STS
SCHEMBL6063814 0.81 CYP19A1 (0.38) CYP19A1CTSLCYP11B1CYP11B2
SCHEMBL8323116 0.81 CYP19A1 (0.39) CYP19A1STSCTSL
SCHEMBL27287580 0.81 CYP11B1 (0.44) CYP19A1STSCTSLCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed