SCHEMBL8329447

SCHEMBL8329447

CCOC(=O)c1cc2cc(NC(=O)CC(C)(C)C)ccc2n1CC1CCCCC1

nearest known ligand 0.71

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 17/20 0.71
ALDH1A1 P00352 1/20 0.41
KCNQ3 O43525 1/20 0.40
KCNQ2 O43526 1/20 0.40
KCNQ4 P56696 1/20 0.40
KCNQ5 Q9NR82 1/20 0.40
RORC P51449 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8363443 0.88 ECE1 (0.81) ECE1KCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL6002242 0.81 ECE1 (0.47) ECE1ALDH1A1RORC
SCHEMBL6019060 0.77 ECE1 (0.74) ECE1
SCHEMBL8363856 0.76 ECE1 (0.49) ECE1KCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL6019583 0.76 ECE1 (0.73) ECE1ALDH1A1
SCHEMBL6019258 0.76 ECE1 (0.75) ECE1
SCHEMBL16473015 0.75 NOD2 (0.55) ALDH1A1
SCHEMBL28305009 0.72 NOD2 (0.66) ALDH1A1
SCHEMBL2433031 0.70 AR (0.51) ALDH1A1
SCHEMBL16747379 0.70 F11 (0.40) ECE1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056768-A2 USE OF SUBSTITUTED 2,5-DIAMIDOINDOLES FOR THE TREATMENT OF UROLOGICAL DISEASES BAYER HEALTHCARE AG (DE) 2004-07-08 WO disclosed
WO-2003028719-A1 SUBSTITUTED 2,5-DIAMIDOINDOLES AS ECE INHIBITORS FOR THE TREATMENT OF CARDIOVASCULAR DISEASES BAYER HEALTHCARE AG (DE) 2003-04-10 WO disclosed