SCHEMBL8329627

SCHEMBL8329627

O=[N+]([O-])c1ccc(CN2CCCCCCCCCCC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.71
ALDH1A1 P00352 1/20 0.69
LMNA P02545 1/20 0.69
MAPT P10636 1/20 0.69
KCNJ1 P48048 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
HRH3 Q9Y5N1 3/20 0.68
CASP1 P29466 1/20 0.60
CASP4 P49662 1/20 0.60
CASP5 P51878 1/20 0.60
CCR2 P41597 1/20 0.60
HRH4 Q9H3N8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1805498 1.00 KDM4E (0.71) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL3143167 1.00 KDM4E (0.71) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL2206628 0.98 KDM4E (0.73) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL3156886 0.95 KDM4E (0.73) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL4021524 0.85 CXCR4 (0.65) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL20640309 0.85 TRPV6 (0.62) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL9621043 0.84 CXCR4 (0.67) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL23832519 0.84 KDM4E (0.69) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL5626457 0.84 ALDH1A1 (0.74) KDM4EALDH1A1LMNAMAPTKCNJ1
SCHEMBL7514453 0.83 KDM4E (0.67) KDM4EALDH1A1LMNAMAPTKCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736035-A4 PRETARGETING METHODS AND COMPOUNDS NEORX CORP (US) 1999-09-01 EP disclosed
US-5847121-A Production of nitro-benzyl-dota via direct peptide cyclization NEORX CORPORATION (US) 1998-12-08 US disclosed
EP-0736035-A1 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1996-10-09 EP disclosed
US-5541287-A DIAGNOSIS USING CYCLIC TRIPEPTIDES WITH NITROBENZYL 1,4,7,10-TETRAAZACYCLODODECANE-N,N*,N**,N***TETRAACETIC ACID BIOTIN CONJUGATE FORMED BY ALKYLATION AND MULTISTAGE PROCESS NEORX CORPORATION (US) 1996-07-30 US disclosed
WO-1995015335-A2 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1995-06-08 WO disclosed
EP-0296522-A2 Functionalized polyamine chelants and rhodium complexes thereof and process for their preparation THE DOW CHEMICAL COMPANY (US) 1988-12-28 EP disclosed