SCHEMBL8329835

SCHEMBL8329835

CN(c1c(C#N)/c(=N/C(=O)Nc2ccccc2)n(C)c(=S)n1-c1ccccc1)C1CN(Cc2ccc(Cl)cc2)CCO1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
FAAH O00519 3/20 0.34
GRIN2B Q13224 1/20 0.33
HIF1A Q16665 1/20 0.32
EPAS1 Q99814 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
CNR2 P34972 2/20 0.32
PKM P14618 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329839 0.84 DRD4 (0.41) DRD4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8327397 0.78 GRIN2B (0.38) DRD4CYP1A2CYP3A4CYP2C9GRIN2B
SCHEMBL8328089 0.78 DRD4 (0.41) DRD4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8328088 0.78 DRD4 (0.41) DRD4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8329877 0.74 DRD4 (0.43) DRD4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8329875 0.74 DRD4 (0.43) DRD4CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8329130 0.71 DRD4 (0.41) DRD4ALDH1A1TSHRCNR2HTT
SCHEMBL8327547 0.71 DRD4 (0.40) DRD4CYP1A2CYP3A4CYP2C9FAAH
SCHEMBL8327545 0.71 DRD4 (0.40) DRD4CYP1A2CYP3A4CYP2C9FAAH
SCHEMBL8325128 0.70 DRD4 (0.41) DRD4ALDH1A1TSHRCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed