SCHEMBL8330293

SCHEMBL8330293

Cc1c2cccn(CC(=O)c3ccccc3)c-2nc1-c1ccc(C(=O)OC(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.46
CD274 Q9NZQ7 1/20 0.46
ALDH1A1 P00352 5/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
GRM1 Q13255 1/20 0.39
GABRA5 P31644 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
BCL2 P10415 1/20 0.37
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
ALDH1A2 O94788 1/20 0.35
ALDH1A3 P47895 1/20 0.35
CA12 O43570 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327343 0.89 ALDH1A1 (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL8328480 0.86 MEN1 (0.42) SMN1; SMN2MEN1KMT2APOLBL3MBTL1
SCHEMBL8326687 0.85 SRC (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL8322914 0.83 NPC1 (0.46) ALDH1A1NPC1RAB9AMAPTL3MBTL1
SCHEMBL8327249 0.83 GSK3B (0.42) RAB9ALMNAHTTMEN1KMT2A
SCHEMBL8329544 0.75 KMT2A (0.45) ALDH1A1RAB9ASMN1; SMN2LMNAHTT
Hydrochloric Acid SCHEMBL8329003 0.74 KMT2A (0.44) ALDH1A1RAB9ASMN1; SMN2LMNAHTT
SCHEMBL8326905 0.73 POLB (0.50) ALDH1A1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL8328201 0.73 PLAA (0.39) ALDH1A1SMN1; SMN2LMNAHTTMEN1
Bromide SCHEMBL8327071 0.72 PLAA (0.38) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509974-B1 Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof ASTRA AB (SE) 1999-01-13 EP disclosed
US-5439917-A Phenyl-pyrrolo(2,3-b)pyridine antisecretory agent of gastric acid; adenosine triphosphatase enzyme inhibitor AKTIEBOLAGET ASTRA (SE) 1995-08-08 US disclosed
EP-0580616-A1 NEW ACTIVE COMPOUNDS Astra Aktiebolag (SE) 1994-02-02 EP disclosed
EP-0509974-A1 Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof Astra Aktiebolag (SE) 1992-10-21 EP disclosed
WO-1992017477-A1 NEW ACTIVE COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1992-10-15 WO disclosed