SCHEMBL8330901

SCHEMBL8330901

OCCOCCNCc1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.53
KCNH3 Q9ULD8 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
ALDH1A1 P00352 2/20 0.47
SCN8A Q9UQD0 1/20 0.47
MPO P05164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 2/20 0.46
LTA4H P09960 1/20 0.45
EPHX2 P34913 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
MITF O75030 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1625040 0.91 ALDH1A1 (0.49) L3MBTL1ALDH1A1KDM4ELMNAMAPK1
SCHEMBL23648099 0.83 APP (0.44) L3MBTL1ALDH1A1KDM4ELMNAMAPK1
SCHEMBL4591762 0.83 CYP1A2 (0.47) ALDH1A1KDM4ELMNACYP2D6CYP2C19
SCHEMBL4406338 0.82 DRD4 (0.58) CHRM2ALDH1A1KDM4ELMNAMAPK1
SCHEMBL4599034 0.81 CHRM2 (0.64) CHRM2L3MBTL1ALDH1A1MPOKDM4E
SCHEMBL6660880 0.81 DRD4 (0.56) CHRM2ALDH1A1KDM4ELMNAMAPK1
SCHEMBL7497061 0.81 CHRM2 (0.55) CHRM2L3MBTL1ALDH1A1SCN8AMPO
SCHEMBL25173760 0.79 SMN1; SMN2 (0.65) L3MBTL1ALDH1A1KDM4ELMNA
SCHEMBL25419906 0.79 SMN1; SMN2 (0.46) ALDH1A1KDM4ELMNAHDAC1CYP2D6
SCHEMBL17664562 0.79 APP (0.51) L3MBTL1ALDH1A1KDM4ELMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed