SCHEMBL8332964

SCHEMBL8332964

CC1(C)CCOc2ccc(C/C=C\CO)cc21

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 1/20 0.46
CYP26B1 Q9NR63 1/20 0.46
RARA P10276 6/20 0.44
RARB P10826 5/20 0.44
RARG P13631 5/20 0.44
RXRA P19793 4/20 0.41
SSTR5 P35346 2/20 0.40
MAP3K14 Q99558 1/20 0.37
HNF4A P41235 1/20 0.36
AKR1B1 P15121 2/20 0.35
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3998188 0.83 CYP26A1 (0.49) CYP26A1CYP26B1RARARARBRARG
SCHEMBL2246604 0.83 CYP26A1 (0.51) CYP26A1CYP26B1RARARARBRARG
SCHEMBL8773454 0.80 CYP26A1 (0.49) CYP26A1CYP26B1RARARARBRARG
SCHEMBL8330612 0.80 RARA (0.58) CYP26A1CYP26B1RARARARBRARG
SCHEMBL2243072 0.77 CYP26A1 (0.48) CYP26A1CYP26B1RARARARBRARG
SCHEMBL12348759 0.77 CYP26A1 (0.48) CYP26A1CYP26B1RARARARBRARG
SCHEMBL6146899 0.75 CYP26A1 (0.69) CYP26A1CYP26B1RARARARBRARG
SCHEMBL10959891 0.74 CYP26A1 (0.46) CYP26A1CYP26B1RARARARBRARG
SCHEMBL8698629 0.74 RARA (0.55) CYP26A1CYP26B1RARARARBRARG
SCHEMBL8328531 0.73 RARA (0.44) CYP26A1CYP26B1RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5917082-A 2,4-pentadienoic acid derivatives having retinoid-like biological activity ALLERGAN SALES, INC. (US) 1999-06-29 US disclosed
US-5886005-A 4-Aza-19-norandrostane derivatives MERCK & CO., INC. (US) 1999-03-23 US disclosed
US-5817836-A 2,4-pentadienoic acid derivatives having retinoid-like biological activity ALLERGAN (US) 1998-10-06 US disclosed
US-5780647-A 2,4-Pentadienoic acid derivatives having retinoid-like biological activity ALLERGAN (US) 1998-07-14 US disclosed
EP-0804205-A4 4-AZA-19-NORANDROSTANE DERIVATIVES MERCK & CO INC (US) 1998-05-20 EP disclosed
EP-0804205-A1 4-AZA-19-NORANDROSTANE DERIVATIVES Merck & Co., Inc. (US) 1997-11-05 EP disclosed
US-5675033-A FOR TREATMENT OF SKIN DISORDERS ALLERGAN (US) 1997-10-07 US disclosed
WO-1996022100-A1 4-AZA-19-NORANDROSTANE DERIVATIVES MERCK & CO., INC. (US) 1996-07-25 WO disclosed